99% Tianeptine konutai tote CAS 30123-17-2
Whakatakotoranga
ITEM | Paerewa | HUA |
Te ahua | Ma ki te paura kowhai | Te paura tioata ma |
Wairewa | Ka whakarewa noa ki te wai me te mewaro me te dichloromethane | Ka rite |
Tautuhinga | Na IR, Kia rite ki te paerewa mahi | Ka rite |
(2) Ka hoatu tauhohenga o te konutai | Ka rite | |
Nga poke A | ≤0.1% | Kaore i kitea |
Pūhui pātahi | Tetahi Max kotahi poke≤0.1% | 0.060% |
Tapeke poke≤0.4% | 0.36% | |
Wairewa Toenga (GC) | Acetidin≤ 0.5% | ND |
Dichloromethane≤ 0.06% | ND | |
Mewaro≤ 0.3% | ND | |
Acetone≤ 0.5% | 0.29% | |
Acetonitrile≤0.041% | 0.022% | |
Ewaro≤0.5% | ND | |
N, N-dimethylformamide≤0.088% | ND | |
Wai | ≤ 5.0% | 3.8% |
Whakamātautau (HPLC) | 99.0%-101.0%(I runga anhydrousbasis) | 99.70% |
Taupānga
Tianeptine konutaite totehe antidepressant tricyclic.He rereke te tikanga o te mahi whakaahuru i te ahua o nga raau taero tricyclic tuku iho.Ka taea e ia te whakanui ake i te reuptake o 5-HT i roto i te kohanga synaptic.Nga paanga o te HT neuronal conduction.Kaore he hononga mo te choline me nga kaiwhakawhiwhi adrenergic.He rite tonu te kaha o te whakamarumaru ki te tricyclics, engari he pai ake te manawanui i tera o te tricyclics.Mo te maimoatanga o te ngawari, te ngawari, te pouri nui ranei, te neurogenic me te reactive depression, te awangawanga me te pouri ki te tinana, ina koa te mamae o te kopu, me te awangawanga me te pouri o nga turoro e whakawhirinaki ana ki te waipiro i te wa e tango ana.